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Product Name | UNC0642 |
Description | A selective inhibitor of G9a and GLP methyltransferases that competitively inhibits binding of H3K9 substrates with a Ki = 3.7 nM; reduces H3K9 dimethylation levels in MDA-MB-231 and PANC-1 cells (IC50s = 110 and 40 nM, respectively); displays improved pharmacokinetic properties relative to UNC0638 |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | methylation histone methyltransferase G9a G9a-like protein GLP inhibitor H3K9 biochemical chromatin research modification gene regulation epigenetic inhibit UNC-0642 selective dimethylation MDA-MB-231 PANC-1 cells UNC-0638 pharmacokinetic SGC structural genomic consortium |
Gene, Accession, CAS # | CAS: 1481677-78-4 |
Catalog # | 14604-1 |
Price | $62.00 |
Order / More Info | UNC0642 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |